Start Date

2018

Description

Indolizines are a versatile heterocyclic core found frequently in pharmaceutical targets for a wide range of therapeutic areas, including anti-tumor treatments,1 an inhibitor of Lp-PLA2, 2 and antagonists of CRTH2, 3 (Figure 1). As such, efficient synthetic methods, with broad substrate scope, for the preparation of substituted indolizines are of significant importance

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Jan 1st, 12:00 AM

Synthesis of Trisubstituted Indolizines: Substitution, on the Pyridine Ring

Indolizines are a versatile heterocyclic core found frequently in pharmaceutical targets for a wide range of therapeutic areas, including anti-tumor treatments,1 an inhibitor of Lp-PLA2, 2 and antagonists of CRTH2, 3 (Figure 1). As such, efficient synthetic methods, with broad substrate scope, for the preparation of substituted indolizines are of significant importance